Apalutamide Intermediates

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Product name: N-Boc-1-aminocyclobutanecarboxylic acid

Alias: N-BOC-1-AMINOCYCLOBUTANECARBOXYLICACID;1-AMINOCYCLOBUTYL-1-CARBOXYLICACID,N-BOCPROTECTED;1-(BOC-AMINO) CYCLOBUTANECARBOXYLICACID;1-N-BOC-AMINO-CYCLOBUTANECARBOXYLICACID;1-(TERT-BUTYLOXYCARBONYL-AMINO)-CYCLOBUTYL-1-CARBOXYLICACID; 1-(TERT-BUTYLOXYCARBONYL-AMINO)-1-(BOC-AMINO)-1-(BOC-AMINO) Aminocyclobutane-1-carboxylicacid,N-BOCprotected;Boc-1-amino-1-cyclobutanecarboxylicacid,97.5%;1-(TERT-BUTYLOXYCARBONYL-AMINO) -CYCLOBUTYL-1-CARBOXYLICACID CYCLOBUTANECARBOXYLICACID

CAS No. 120728-10-1

Molecular Formula: C10H17NO4

Molecular weight: 215.25

Properties: white crystalline powder

Melting point: 129-133°C(lit.)

Boiling point: 362.1±21.0°C(Predicted)

Density: 1.18±0.1g/cm3(Predicted)

Storage conditions: Keepindarkplace,Sealedindry,RoomTemperature

Solubility: Soluble in methanol

Acidity coefficient: (pKa)4.14±0.20(Predicted)

Form: Powder

Color: white to light brown

Application: Used as pharmaceutical intermediate of Apatamide.

Product specification: 1kg/drum, 2kg/drum, 5kg/drum, 10kg/drum, 15kg/drum, 20kg/drum, 25kg/drum, etc., and can be separately subcontracted according to customers' requirements.

Price: Price is for reference only, call us for one-to-one quotation.

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Upstream raw materials: 1-aminocyclobutanecarboxylic acid 5,7-Diaza-spiro[3.4]octane-6,8-dione BOC-1-aminocyclobutanecarboxylic acid ethyl ester Ethyl 1-bromocyclobutanecarboxylate

Downstream products: BOC-1-aminocyclobutanecarbonitrile

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Molecular structure：